Receptor-Ligand結合分析實驗


 非放射性接合子 (Non-Radiolabeled Ligands)

 本公司提供來自英國Ascent Scientific公司的多種優質非放射線標定的接合子(Ligand)產品,如下表所示。
 如果您在此表找不到適當的Ligand,煩請聯絡本公司客服部為您尋找。


Ligand Purity Ref. No. Pack Size
ACEA >98% Asc-096 5mg
Potent, selective CB1 agonist 25mg
  100mg
AF-DX 116 >99% Asc-152 10mg
M2 antagonist 50mg
AM 251 >99% Asc-088 10mg
CB1 receptor antagonist / inverse agonist 50mg
AM404 >99% Asc-095 10mg
Anandamide transport inhibitor 50mg
Aminoguanidine hydrochloride >98% Asc-123 100mg
NOS inhibitor
4-Aminopyridine >99% Asc-122 100mg
K+ channel blocker
AMN082 dihydrochloride >99% Asc-011 10mg
mGlu7 agonist 50mg
(RS)-AMPA >99% Asc-130 10mg
AMPA agonist 50mg
(S)-AMPA >98% Asc-005 5mg
AMPA agonist 10mg
  50mg
Anandamide >98% Asc-087 5mg
Endogenous cannabinoid 25mg
(±)-Anatoxin A fumarate >98% Asc-013 1mg
Potent nicotinic agonist
DL-AP4 >99% Asc-001 100mg
NMDA receptor antagonist 1g
L-AP4 >99% Asc-002 10mg
Selective group III mGlu agonist 50mg
D-AP5 >99% Asc-003 10mg
NMDA glutamate site antagonist 50mg
  100mg
DL-AP5 >99% Asc-004 10mg
NMDA glutamate site antagonist 50mg
2-APB >98% Asc-124 100mg
Ca2+ release modulator
Apigenin >98% Asc-141 10mg
Anticancer agent 50mg
AQ-RA 741 >99% Asc-151 10mg
M2 antagonist 50mg
(RS)-Baclofen >99% Asc-149 1g
GABAB agonist
(+)-Bicuculline >98% Asc-107 50mg
GABAA antagonist.
(-)-Bicuculline methiodide >98% Asc-108 10mg
GABAA antagonist. 50mg
(-)-Bicuculline methobromide >98% Asc-109 10mg
GABAA antagonist. 50mg
(-)-Bicuculline methochloride >98% Asc-110 10mg
GABAA antagonist. 50mg
Nor-Binaltorphimine >98% Asc-078 10mg
Potent and selective k opioid receptor antagonist 50mg
Camptothecin >98% Asc-115 50mg
DNA topoisomerase inhibitor 250mg
Capsazepine >99% Asc-025 10mg
VR1 antagonist 50mg
CGP 37157 >99% Asc-012 10mg
Na+-Ca2+ exchange inhibitor 50mg
CGP 37849 >99% Asc-127 10mg
Competitive NMDA antagonist 50mg
CGP 39551 >99% Asc-128 10mg
Competitive NMDA antagonist 50mg
2-Chloroadenosine >98% Asc-037 10mg
Adenosine agonist 50mg
  250mg
7-Chlorokynurenic acid >99% Asc-024 10mg
NMDA receptor glycine site antagonist 50mg
(S)-5-Chlorowillardiine >98% Asc-062 10mg
AMPA / Kainate agonist 50mg
(RS)-CHPG >98% Asc-039 10mg
Selective mGlu5 agonist 50mg
Citalopram >98% Asc-133 25mg
5HT reuptake inhibitor 100mg
Clozapine >98.5% Asc-019 50mg
Atypical antipsychotic 500mg
CNQX >99% Asc-017 10mg
AMPA / kainate antagonist 25mg
  50mg
CNQX disodium salt >99% Asc-044 10mg
AMPA / kainate antagonist (water soluble) 50mg
CPCCOEt >98% Asc-060 10mg
Selective, non-competitive mGlu1 antagonist 50mg
Cycloheximide >98% Asc-093 100mg
Protein synthesis inhibitor 1g
D-Cycloserine >99% Asc-121 50mg
NMDA glycine site agonist 250mg
Cyclosporin A >99% Asc-114 25mg
PP2B inhibitor 100mg
  500mg
Cyclothiazide >98% Asc-061 10mg
AMPA receptor desensitisation inhibitor 50mg
4-DAMP >98% Asc-144 25mg
Muscarinic receptor antagonist 100mg
(S)-3,4-DCPG >99% Asc-006 10mg
mGlu8a agonist 50mg
N-Desmethyl clozapine >99% Asc-026 10mg
Clozapine metabolite. M1 agonist. 50mg
Desmethyl YM298198 hydrochloride >99% Asc-016 10mg
Analogue of mGlu1 antagonist YM298198 50mg
(R,S)-3,5-DHPG >98% Asc-020 10mg
Group I mGlu receptor agonist 50mg
(S)-3,5-DHPG >99% Asc-007 5mg
Selective group I mGlu agonist. 10mg
5,7-Dichlorokynurenic acid >99% Asc-023 10mg
NMDA receptor glycine site antagonist 50mg
  100mg
Dihydrokainic acid >99% Asc-066 10mg
EAAT2 inhibitor 50mg
DNQX >99% Asc-018 10mg
AMPA / kainate antagonist 50mg
E-4031 dihydrochloride >99% Asc-158 10mg
HERG K+ channel blocker 50mg
FCCP >99% Asc-081 10mg
Mitochondrial oxidative phosphorylation inhibitor 50mg
Fenobam >99% Asc-034 10mg
Selective, potent, orally active mGlu5 antagonist 50mg
(S)-5-Fluorowillardiine >99% Asc-036 10mg
Potent, selective AMPA agonist 50mg
Fluoxetine hydrochloride >99% Asc-077 10mg
5HT reuptake inhibitor 50mg
Forskolin >98% Asc-058 10mg
Adenylate cyclase activator 50mg
  100mg
Genistein >99% Asc-112 10mg
Protein tyrosine kinase inhibitor. Anticancer agent. 50mg
  100mg
L-Glutamate >99% Asc-049 1g
Excitatory neurotransmitter 2.5g
Glycine >99% Asc-050 100mg
Inhibitory neurotransmitter 1g
Granisetron >99% Asc-125 50mg
5HT3 antagonist 250mg
Haloperidol >99% Asc-080 100mg
D2 antagonist
Herkinorin >98% Asc-147 1mg
Non-internalising μ opioid agonist
Ibotenic acid >98% Asc-041 5mg
Excitotoxic agonist 25mg
ICI 182,780 >99% Asc-131 10mg
Estrogen receptor antagonist 50mg
Ifenprodil >99% Asc-111 10mg
NR2B-preferring NMDA antagonist 50mg
Ionomycin Ca2+ Salt >99% Asc-116 1mg
Ca2+ ionophore. 5mg
Isradipine >98% Asc-142 10mg
L-type Ca2+ channel blocker 50mg
Kainic acid >99% Asc-100 10mg
Prototypic kainate receptor agonist 50mg
Ketanserin tartrate >98% Asc-132 50mg
Selective 5HT2 antagonist. 250mg
Kynurenic acid >98% Asc-064 1g
Endogenous ionotropic / nicotinic antagonist
(R,S)-MCPG >99% Asc-033 10mg
Group I /II metabotropic glutamate antagonist 50mg
(S)-MCPG >98% Asc-059 10mg
Group I / II mGlu antagonist 50mg
(R)-(-)-α-Methylhistamine dihydrobromide >98% Asc-053 10mg
Potent, selective H3 agonist 50mg
N-Methyllidocaine iodide >99% Asc-119 10mg
Anti-arrthymic 50mg
Methyllycaconitine citrate >98% Asc-072 5mg
α7- nicotinic receptor antagonist 25mg
Mirtazepine >99% Asc-068 10mg
Antidepressant. α2, 5HT2, 5HT3 antagonist. 50mg
(-)-MK 801 maleate >99% Asc-028 10mg
Non competitive NMDA antagonist; less active enantiomer 50mg
(+)-MK 801 maleate >99% Asc-027 10mg
Non-competitive NMDA antagonist 50mg
MPEP hydrochloride >99% Asc-008 10mg
Potent, selective mGlu5 antagonist 50mg
MTEP hydrochloride >99% Asc-035 10mg
Potent, selective mGlu5 antagonist 50mg
Muscimol >99% Asc-094 5mg
Potent, selective GABAA agonist. 10mg
  50mg
NADA >98% Asc-099 5mg
Endogenous CB1 / TRPV1 agonist 25mg
Naloxone hydrochloride >98% Asc-074 100mg
Opioid antagonist 250mg
Naltrexone hydrochloride >98% Asc-075 100mg
Opioid antagonist 250mg
NBQX >99% Asc-045 10mg
AMPA / kainate antagonist 50mg
NBQX disodium salt >99% Asc-046 10mg
AMPA / kainate antagonist; water soluble 50mg
Nicotinic acid >98% Asc-145 10g
Antidyslipidemic agent
Nifedipine >99% Asc-135 250mg
L-type Ca2+ channel blocker 1g
Nimodipine >98% Asc-138 100mg
L-type Ca2+ channel blocker 500mg
Nitrendipine >98% Asc-139 100mg
L-type Ca2+ channel blocker 500mg
(S)-5-Nitrowillardiine >98% Asc-063 10mg
AMPA / Kainate agonist 50mg
NMDA >98% Asc-052 50mg
Excitotoxic amino acid 100mg
  500mg
Nociceptin >95% Asc-070 1mg
ORL1 agonist 5
Obestatin >95% Asc-071 1mg
Endgoenous peptide involved in feeding
ODQ >99% Asc-022 10mg
Selective, potent inhibitor of NO-sensitive guanylyl cyclase 50mg
Ondansetron >98% Asc-134 10mg
Selective 5HT3 antagonist. 50mg
Paclitaxel >98% Asc-143 10mg
Anticancer agent 50mg
Paroxetine hydrochloride >99% Asc-069 10mg
5HT uptake inhibitor 50mg
2,3 cis-Piperidine dicarboxylic acid >98% Asc-038 50mg
ionotropic receptor antagonist 250mg
PHCCC >98% Asc-043 10mg
Selective allosteric potentiator at mGlu4 50mg
Phospho-Glycogen Synthase Peptide-2 >99% Asc-079 0.5mg
1mg
Pirenzepine dihydrochloride >99% Asc-153 100mg
M1 antagonist 500mg
PPADS   Asc-009 10mg
P2 purinergic receptor antagonist. 50mg
  250mg
cis-PPDA >98% Asc-047 10mg
NR2C/NR2D NMDA antagonist 50mg
PPT >99% Asc-161 10mg
Subtype selective ERα agonist 50mg
Quisqualic acid >99% Asc-010 5mg
Group I mGlu agonist. AMPA agonist 10mg
  50mg
QX-222 >99% Asc-126 10mg
Na+ channel blocker 50mg
QX-314 bromide >99% Asc-117 50mg
Na+ channel blocker 100mg
QX-314 chloride >99% Asc-118 50mg
Na+ channel blocker
Reboxetine mesylate >99% Asc-157 10mg
Noradrenaline reuptake inhibitor 50mg
(R,S)-Rolipram >99% Asc-029 10mg
Selective PDE4 inhibitor 50mg
(R)-(-)-Rolipram >98.5% Asc-031 10mg
Selective PDE4 inhibitor 50mg
(S)-(+)-Rolipram >99% Asc-030 10mg
PDE4 inhibitor; less active enantiomer 50mg
Ryanodine >98% Asc-083 1mg
Ca2+ release modulator
Salvinorin A >99% Asc-084 1mg
Potent κ agonist
D-Serine >99% Asc-048 1g
Endogenous NMDA receptor co-agonist 5g
SL 327 >99% Asc-082 10mg
MEK inhibitor 25mg
SNAP   Asc-014 10mg
NO donor 50mg
SP600125 >98% Asc-065 10mg
JNK inhibitor 50mg
Spermidine hydrochloride >99% Asc-057 100mg
Endogenous polyamine. nNOS inhibitor.
Spermine >99% Asc-051 100mg
Endogenous polyamine 1g
SR95531 >98% Asc-042 10mg
GABAA antagonist 50mg
Staurosporine >98% Asc-056 0.1mg
Protein kinase inhibitor 0.5mg
Tetrodotoxin >98% Asc-054 1mg
Na+ channel blocker
Tetrodotoxin citrate >98% Asc-055 1mg
Na+ channel blocker; water-soluble
(+/-)-Thalidomide >99% Asc-032 100mg
Immunomodulator and anticancer agent
Thioperamide maleate >99% Asc-021 10mg
Potent, selective H3 antagonist 50mg
Tropisetron hydrochloride >99% Asc-156 10mg
5-HT3 antagonist 50mg
(+)-Tubocurarine >99% Asc-073 10mg
ACh receptor antagonist 50mg
Verapamil hydrochloride >99% Asc-140 1g
L-type Ca2+ channel blocker
(S)-Willardiine >98% Asc-040 10mg
AMPA / kainate receptor agonist 50mg
Wortmannin >98% Asc-148 1mg
PI3-kinase inhibitor 5mg
XE-991 dihydrochloride >99% Asc-089 10mg
Potent, selective KCNQ channel blocker; blocks M current 50mg
Y-27632 dihydrochloride >99% Asc-129 1mg
Selective Rho kinase inhibitor 10mg
  50mg
YM298198 hydrochloride >99% Asc-015 10mg
Potent, selective mGlu1 antagonist 50mg
ZD7288 >98% Asc-102 10mg
Sino-atrial node function modulator 50mg
Zopiclone >98% Asc-076 10mg
Benzodiazepine agonist 50mg